SCHEMBL19852298

SCHEMBL19852298

COc1ccccc1OC1CCN(CC2c3ccc(CC4(C)Cc5ccccc5C4CN4CCC(Oc5ccccc5OC)CC4)cc3CC2C)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.35
HTR7 P34969 5/20 0.35
SIGMAR1 Q99720 2/20 0.34
HTR1A P08908 2/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
MAPK1 P28482 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
ATM Q13315 1/20 0.32
HTR2C P28335 3/20 0.32
SMPD1 P17405 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21071614 0.81 HTR7 (0.45) HTR7SIGMAR1HTR1AMEN1KMT2A
SCHEMBL21145387 0.77 SLC6A2 (0.42) OPRM1HTR7SIGMAR1HTR1AMEN1
SCHEMBL19852349 0.67 SIGMAR1 (0.52) HTR7SIGMAR1HTR1AHTR2CDRD2
SCHEMBL19852462 0.66 OPRM1 (0.40) OPRM1HTR7HTR1AMEN1KMT2A
SCHEMBL19852300 0.66 HTR7 (0.47) HTR7SIGMAR1HTR1AMEN1KMT2A
SCHEMBL19852152 0.65 PDE4A (0.43) HTR7MEN1KMT2APDE4APDE4B
SCHEMBL25619737 0.64 LMNA (0.50) SIGMAR1HTR1ADRD2
SCHEMBL19852460 0.60 KCNH2 (0.46) SIGMAR1HTR1AMEN1KMT2AADRA1D
SCHEMBL19374778 0.60 SMN1; SMN2 (0.52) OPRM1HTR1AMEN1KMT2ACYP2D6
SCHEMBL19852164 0.60 SIGMAR1 (0.44) HTR7SIGMAR1HTR1AHTR2CDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026371-A1 DUAL NAV1.2/5HT2A INHIBITORS FOR TREATING CNS DISORDERS SUNOVION PHARMACEUTICALS INC. (US) 2018-02-08 WO disclosed