SCHEMBL19853420

SCHEMBL19853420

CNCCNOCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
L3MBTL1 Q9Y468 3/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SIGMAR1 Q99720 2/20 0.46
HRAS P01112 1/20 0.45
CYP3A4 P08684 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 2/20 0.43
TMEM97 Q5BJF2 1/20 0.43
CARM1 Q86X55 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
PRMT8 Q9NR22 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
HTR1B P28222 2/20 0.42
HTR1D P28221 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1240611 0.82 HRAS (0.46) ATMTAAR1SIGMAR1HRASTSHR
SCHEMBL437919 0.79 MAOA (0.48) L3MBTL1SIGMAR1HRASTSHRNPC1
SCHEMBL1829762 0.79 NPC1 (0.50) ATMTAAR1L3MBTL1SIGMAR1HRAS
SCHEMBL19853459 0.78 MEN1 (0.65) MEN1KMT2ASIGMAR1HRASMAPT
SCHEMBL16352091 0.78 NPC1 (0.45) ATMTAAR1HRASTSHRNPC1
SCHEMBL8150074 0.78 HRAS (0.50) HRASTSHRNPC1RAB9AIDO1
Hydrochloric Acid SCHEMBL6436425 0.78 GAA (0.50) ATMTAAR1L3MBTL1MEN1KMT2A
SCHEMBL10948517 0.78 NPC1 (0.47) TAAR1HRASCYP3A4TSHRNPC1
SCHEMBL17805686 0.78 HRAS (0.46) MEN1KMT2AHRASTSHRNPC1
SCHEMBL19853411 0.77 TAAR1 (0.48) TAAR1SIGMAR1HRASTSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026792-A1 SPIRO-LACTAM AND BIS-SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed