SCHEMBL19853411

SCHEMBL19853411

CN(C)CCNOCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.48
SIGMAR1 Q99720 1/20 0.43
HRAS P01112 1/20 0.42
TSHR P16473 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LTA4H P09960 2/20 0.41
EGFR P00533 2/20 0.41
LYPLA1 O75608 1/20 0.40
LYPLA2 O95372 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DRD2 P14416 1/20 0.39
DRD1 P21728 1/20 0.39
DRD4 P21917 1/20 0.39
DRD5 P21918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1240611 0.79 HRAS (0.46) TAAR1SIGMAR1HRASTSHRALDH1A1
SCHEMBL19853420 0.77 ATM (0.52) TAAR1SIGMAR1HRASTSHRLTA4H
SCHEMBL437919 0.76 MAOA (0.48) SIGMAR1HRASTSHRNPC1RAB9A
SCHEMBL1829762 0.76 NPC1 (0.50) TAAR1SIGMAR1HRASTSHRALDH1A1
SCHEMBL21362339 0.75 FOLH1 (0.39) HRASALDH1A1NPC1RAB9A
SCHEMBL10948517 0.75 NPC1 (0.47) TAAR1HRASTSHRALDH1A1NPC1
SCHEMBL8150074 0.75 HRAS (0.50) HRASTSHRLTA4HNPC1RAB9A
SCHEMBL17805686 0.75 HRAS (0.46) HRASTSHRALDH1A1NPC1RAB9A
Hydrochloric Acid SCHEMBL6436425 0.75 GAA (0.50) TAAR1SIGMAR1HRASTSHRALDH1A1
Hydrochloric Acid SCHEMBL7870266 0.74 SIGMAR1 (0.44) SIGMAR1HRASTSHRALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026792-A1 SPIRO-LACTAM AND BIS-SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed