SCHEMBL19854301

SCHEMBL19854301

CC(C)CNCNC1CCC2(CC1)CN(CC(N)=O)C2=O

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.30
APEX1 P27695 1/20 0.30
BLM P54132 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21034922 0.92 OPRK1 (0.35) OPRK1APEX1BLM
SCHEMBL19854883 0.79 GRIN2B (0.38) OPRK1
SCHEMBL19853787 0.78 BLM (0.35) APEX1BLM
SCHEMBL19853725 0.77 APEX1 (0.32) APEX1BLM
SCHEMBL19853794 0.76 APEX1 (0.35) APEX1BLM
SCHEMBL19854298 0.74 OPRM1 (0.34) APEX1BLM
SCHEMBL19839384 0.74 BLM (0.39) APEX1BLM
SCHEMBL19853789 0.72 APEX1 (0.47) APEX1BLM
SCHEMBL19853769 0.69 TSHR (0.44) APEX1BLM
SCHEMBL24634181 0.69 GRIN2B (0.41) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026763-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed