SCHEMBL19856942

SCHEMBL19856942

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)c1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.42
PYGL P06737 1/20 0.41
CYP51A1 Q16850 2/20 0.39
STAT6 P42226 1/20 0.39
CCKAR P32238 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
CNR2 P34972 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
ALOX15 P16050 1/20 0.37
CCR1 P32246 1/20 0.37
PDGFRB P09619 1/20 0.37
PDGFRA P16234 1/20 0.37
DRD3 P35462 4/20 0.37
DRD4 P21917 3/20 0.37
KCNH2 Q12809 1/20 0.37
HTR1A P08908 1/20 0.37
DRD1 P21728 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19856943 1.00 DRD2 (0.42) DRD2PYGLCYP51A1STAT6CCKAR
SCHEMBL19856882 0.93 ALOX15 (0.42) DRD2PYGLCYP51A1STAT6HRH4
SCHEMBL19856883 0.93 ALOX15 (0.42) DRD2PYGLCYP51A1STAT6HRH4
SCHEMBL19856896 0.93 PYGL (0.43) DRD2PYGLCYP51A1STAT6HRH4
SCHEMBL19856898 0.93 PYGL (0.43) DRD2PYGLCYP51A1STAT6HRH4
SCHEMBL19856872 0.93 DRD2 (0.41) DRD2PYGLCYP51A1STAT6CCKAR
SCHEMBL19856871 0.93 DRD2 (0.41) DRD2PYGLCYP51A1STAT6CCKAR
SCHEMBL19856954 0.91 DRD2 (0.42) DRD2PYGLCYP51A1STAT6HRH4
SCHEMBL19856955 0.91 DRD2 (0.42) DRD2PYGLCYP51A1STAT6HRH4
SCHEMBL19856916 0.90 CYP51A1 (0.40) DRD2PYGLCYP51A1STAT6CCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925857-B1 USE OF TRPV4 ANTAGONISTS TO AMELIORATE HYDROCEPHALUS AND RELATED MATERIALS AND METHODS UNIV INDIANA RES & TECH CORP (US) 2018-02-14 EP claimed