SCHEMBL19860009

SCHEMBL19860009

Cc1cc(F)ccc1NC(=O)N1CC2CCCC2C1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 8/20 0.58
HDAC1 Q13547 4/20 0.58
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
GRIN2B Q13224 6/20 0.51
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13833393 0.84 HDAC2 (0.65) HDAC2HDAC1GRIN2B
SCHEMBL18079545 0.83 HDAC2 (0.66) HDAC2HDAC1
SCHEMBL19860010 0.82 RAB9A (0.71) HDAC2HDAC1KDM4ELMNANPC1
SCHEMBL30986004 0.81 RAB9A (0.74) HDAC2HDAC1KDM4ELMNANPC1
SCHEMBL14372234 0.77 RAB9A (0.56) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL19860011 0.76 TAS1R3 (0.75) LMNANPC1RAB9AMAPTMAPK1
SCHEMBL13833449 0.75 HDAC2 (0.78) HDAC2HDAC1
SCHEMBL18376433 0.74 HDAC2 (1.00) HDAC2HDAC1
SCHEMBL12432966 0.73 KDM4E (0.64) KDM4ELMNANPC1RAB9AMAPT
SCHEMBL31020925 0.72 HDAC2 (0.63) HDAC2HDAC1GRIN2BMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890172-B2 Inhibitors of histone deacetylase THE BROAD INSTITUTE, INC. (US) 2018-02-13 US disclosed