SCHEMBL19860065

SCHEMBL19860065

O=C(Cc1ccc(F)cc1)Nc1ccc2cnccc2c1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 3/20 0.61
ROCK2 O75116 3/20 0.60
GAA P10253 2/20 0.60
NOTUM Q6P988 4/20 0.55
SMN1; SMN2 Q16637 1/20 0.53
IMPDH2 P12268 3/20 0.53
PRMT3 O60678 2/20 0.53
HDAC1 Q13547 1/20 0.53
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860082 0.89 ROCK1 (0.60) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL24735962 0.87 IMPDH2 (0.69) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL19860106 0.85 ROCK1 (0.57) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL24736084 0.85 ROCK1 (0.61) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL24736559 0.85 IMPDH2 (0.51) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL19860093 0.85 ROCK2 (0.61) ROCK1ROCK2NOTUMSMN1; SMN2IMPDH2
SCHEMBL14625937 0.85 ROCK2 (0.60) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL24736108 0.83 ROCK1 (0.49) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL24736304 0.83 ROCK1 (0.49) ROCK1ROCK2NOTUMIMPDH2PRMT3
SCHEMBL23736265 0.82 NOTUM (0.50) ROCK1ROCK2NOTUMIMPDH2PRMT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed