SCHEMBL19860121

SCHEMBL19860121

O=C(CCNCc1ccc(C(=O)Nc2ccccc2)cc1)Nc1ccc2cnccc2c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 4/20 0.58
PRMT3 O60678 1/20 0.56
NAMPT P43490 7/20 0.52
NOTUM Q6P988 2/20 0.47
ROCK2 O75116 2/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
BLK P51451 1/20 0.46
BTK Q06187 1/20 0.46
HDAC1 Q13547 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860123 0.90 IMPDH2 (0.71) IMPDH2PRMT3NOTUMROCK2
SCHEMBL14124401 0.89 IMPDH2 (0.61) IMPDH2PRMT3NAMPTNOTUMROCK2
SCHEMBL19860122 0.83 IMPDH2 (0.56) IMPDH2PRMT3NOTUMROCK2
SCHEMBL14124404 0.81 HDAC1 (0.62) IMPDH2PRMT3NOTUMNPC1ALDH1A1
SCHEMBL2164137 0.80 PRMT3 (0.69) IMPDH2PRMT3NAMPTNOTUMROCK2
SCHEMBL3111893 0.79 IMPDH2 (0.72) IMPDH2PRMT3NAMPTROCK2MEN1
SCHEMBL2162616 0.79 IMPDH2 (0.70) IMPDH2PRMT3NOTUMROCK2ALDH1A1
SCHEMBL2162460 0.78 KMT2A (0.67) NAMPTROCK2MEN1NPC1ALDH1A1
SCHEMBL4432783 0.77 IMPDH2 (0.65) IMPDH2PRMT3NAMPTROCK2MEN1
SCHEMBL3566775 0.77 PRMT3 (0.72) IMPDH2PRMT3NOTUMROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed