SCHEMBL19860123

SCHEMBL19860123

O=C(CCNCc1ccccc1)Nc1ccc2cnccc2c1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 5/20 0.71
PRMT3 O60678 4/20 0.68
ROCK2 O75116 6/20 0.54
NOTUM Q6P988 4/20 0.54
ROCK1 Q13464 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19860121 0.90 IMPDH2 (0.58) IMPDH2PRMT3ROCK2NOTUM
SCHEMBL19860122 0.89 IMPDH2 (0.56) IMPDH2PRMT3ROCK2NOTUM
SCHEMBL2162616 0.88 IMPDH2 (0.70) IMPDH2PRMT3ROCK2NOTUMROCK1
SCHEMBL3566775 0.87 PRMT3 (0.72) IMPDH2PRMT3ROCK2NOTUMROCK1
SCHEMBL2164137 0.84 PRMT3 (0.69) IMPDH2PRMT3ROCK2NOTUMROCK1
SCHEMBL2162998 0.83 IMPDH2 (1.00) IMPDH2PRMT3ROCK2ROCK1
SCHEMBL24735962 0.83 IMPDH2 (0.69) IMPDH2PRMT3ROCK2NOTUMROCK1
SCHEMBL14124306 0.82 PRMT3 (0.66) IMPDH2PRMT3ROCK2NOTUMROCK1
SCHEMBL19860125 0.81 PRMT3 (0.71) IMPDH2PRMT3ROCK2NOTUMROCK1
SCHEMBL19860124 0.81 IMPDH2 (0.59) IMPDH2PRMT3NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed