SCHEMBL19861608

SCHEMBL19861608

CS(C)(C)CCOCn1ccc2cnc(Cl)cc21

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.37
CDK2 P24941 1/20 0.37
KMT2A Q03164 1/20 0.33
MAP3K5 Q99683 1/20 0.31
CCR9 P51686 1/20 0.30
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16442052 0.90 CDC7 (0.38) CDC7CDK2KMT2AMAP3K5CCR9
SCHEMBL13732447 0.83 DGAT1 (0.39) CDC7CDK2KMT2ACCR9MCL1
SCHEMBL29777185 0.83 DGAT1 (0.39) CDC7CDK2KMT2ACCR9MCL1
SCHEMBL28521488 0.80 CDC7 (0.41) CDC7CDK2KMT2AMAP3K5CCR9
SCHEMBL19861615 0.75 MEN1 (0.33) KMT2A
SCHEMBL23229422 0.74 CXCR3 (0.30)
SCHEMBL28656926 0.74 GRIN2B (0.43) CDC7CDK2KMT2AMCL1
SCHEMBL23915418 0.73 DUT (0.36)
SCHEMBL24805178 0.73 DGAT1 (0.39) CDC7CDK2KMT2ACCR9
SCHEMBL24493506 0.72 HTR2C (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890152-B2 Aminopyrimidine compounds as inhibitors of T790M containing EGFR mutants GENENTECH, INC. (US) 2018-02-13 US disclosed