SCHEMBL19862430

SCHEMBL19862430

CC(C)c1nc(C(=O)O)cc(N2CCNCC2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.43
CASP4 P49662 1/20 0.43
CASP5 P51878 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
GBA1 P04062 2/20 0.42
ADRB1 P08588 1/20 0.42
NCF1 P14598 1/20 0.42
CYP3A4 P08684 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PRKD1 Q15139 1/20 0.40
PRKD2 Q9BZL6 1/20 0.40
ITGA2B P08514 3/20 0.40
HCAR3 P49019 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
IKBKB O14920 1/20 0.39
ITGB3 P05106 1/20 0.39
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16775737 0.89 CASP1 (0.43) CASP1CASP4CASP5KDM4EMEN1
SCHEMBL16785589 0.82 ADRB1 (0.47) CASP1CASP4CASP5KDM4EMEN1
Hydrochloric Acid SCHEMBL5219717 0.81 HRH4 (0.43) MEN1KMT2AHRH4GBA1IKBKB
SCHEMBL19865043 0.79 ITGA2B (0.46) CASP1CASP4CASP5KDM4EMEN1
SCHEMBL25379567 0.77 GBA1 (0.52) CASP1CASP4CASP5KMT2AHRH4
SCHEMBL30306132 0.77 GBA1 (0.52) CASP1CASP4CASP5KMT2AHRH4
SCHEMBL2902905 0.75 HTT (0.54) KDM4EMEN1KMT2AADRB1NCF1
SCHEMBL21044592 0.73 ADRB1 (0.52) KDM4EADRB1NCF1CYP3A4HSD17B10
SCHEMBL5222137 0.73 CKS1B (0.52) HRH4
SCHEMBL30834235 0.70 HRH3 (0.59) HRH4HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180044338-A1 SUBSTITUTED BRIDGED UREA ANALOGS AS SIRTUIN MODULATORS GLAXOSMITHKLINE LLC (US) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180044338-A1 SUBSTITUTED BRIDGED UREA ANALOGS AS SIRTUIN MODULATORS SIRT1, SIRT3, SIRT2 CASP1 356/4885CASP4 725/4885CASP5 600/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.