SCHEMBL19902346

SCHEMBL19902346

CCC(=O)c1ccn(CCC(F)(F)F)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 3/20 0.38
KDM4C Q9H3R0 1/20 0.36
RAB9A P51151 7/20 0.35
NPC1 O15118 6/20 0.35
MEN1 O00255 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.34
POLB P06746 2/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPT P10636 1/20 0.33
CHRNA7 P36544 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454393 0.84 ALDH1A1 (0.38) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL16796408 0.83 SMN1; SMN2 (0.46) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL17438035 0.82 KMT2A (0.52) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL30209674 0.81 CYP1A2 (0.40) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL17452573 0.81 NPC1 (0.36) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL19902313 0.80 ALDH1A1 (0.39) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL28111821 0.79 ALDH1A1 (0.54) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL12535851 0.73 TSHR (0.51) ALDH1A1KMT2ARAB9ANPC1MEN1
SCHEMBL23985340 0.72 DRD2 (0.39) ALDH1A1CYP1A2CYP2D6RAB9ANPC1
SCHEMBL8531702 0.72 CACNA1H (0.55) ALDH1A1KMT2ACYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed