SCHEMBL19902424

SCHEMBL19902424

CCC(=O)c1cnn2cc(CCCN3CCC(F)(F)C3)ccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 3/20 0.35
CDK8 P49336 3/20 0.35
GRM4 Q14833 1/20 0.35
KCNA3 P22001 1/20 0.35
GRM2 Q14416 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
GLS O94925 1/20 0.33
OPRM1 P35372 3/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
OPRD1 P41143 1/20 0.33
KMT2A Q03164 1/20 0.33
KIF11 P52732 1/20 0.32
JAK2 O60674 1/20 0.32
FGFR1 P11362 1/20 0.32
FGFR2 P21802 1/20 0.32
FGFR4 P22455 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454440 0.91 CCNC (0.36) CCNCCDK8GRM4KCNA3GRM2
SCHEMBL17452720 0.88 HTR2A (0.35) CCNCCDK8GRM4GRM2HTR2A
SCHEMBL17454520 0.85 NOS3 (0.38) CCNCCDK8GRM4KCNA3GRM2
SCHEMBL17452719 0.82 HTR2A (0.38) GRM4KCNA3GRM2HRH3HTR2A
SCHEMBL19902683 0.82 HRH3 (0.42) HRH3HTR2AHTR2CALDH1A1
SCHEMBL19902549 0.77 MET (0.38) JAK2
SCHEMBL19675383 0.76 SIGMAR1 (0.38) HRH3
SCHEMBL23889078 0.75 ROCK2 (0.39) ALDH1A1
SCHEMBL19902395 0.74 THRA (0.37) MEN1KMT2A
SCHEMBL17454474 0.74 SIGMAR1 (0.42) HRH3HTR2AHTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed