SCHEMBL19903359

SCHEMBL19903359

FC1CN(Sc2ccc(Br)cc2)C1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
DPP4 P27487 2/20 0.33
CYP2A6 P11509 1/20 0.32
HRH3 Q9Y5N1 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19903254 0.80 MAOA (0.34) MAOAMAOBCYP2A6HRH3
SCHEMBL19903224 0.76 MAOA (0.32) MAOAMAOBHRH3
SCHEMBL20311368 0.72 MAOB (0.38) MAOAMAOBCYP2A6
SCHEMBL19903214 0.72 HPGD (0.39) MAOAMAOBCYP2A6
SCHEMBL19903237 0.71 HPGD (0.38) MAOAMAOBCYP2A6
SCHEMBL19903239 0.68 TSHR (0.37) MAOAMAOBCYP2A6TSHR
SCHEMBL22643093 0.68 ALDH1A1 (0.47) MAOAMAOBHRH3TSHR
SCHEMBL20108604 0.68 KDM4E (0.47) MAOAMAOBCYP2A6
SCHEMBL20108451 0.68 KMT2A (0.49) TSHR
SCHEMBL19903234 0.67 PDK1 (0.38) MAOAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2976341-B1 ACYCLIC CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-02-28 EP disclosed