SCHEMBL19903993

SCHEMBL19903993

C=CC(=O)Oc1ccc(N)cc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.40
ALDH1A1 P00352 4/20 0.39
THRB P10828 4/20 0.38
THRA P10827 1/20 0.38
TYMS P04818 1/20 0.37
CASP1 P29466 2/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 3/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP19A1 P11511 1/20 0.33
GAA P10253 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21141405 0.84 RAB9A (0.42) THRBTHRATYMSTSHRMAPT
SCHEMBL1696567 0.83 THRB (0.47) ALDH1A1THRBTHRATYMSMAPT
SCHEMBL30593911 0.83 L3MBTL1 (0.47) ALDH1A1THRBTHRATYMSMAPT
SCHEMBL39820 0.83 L3MBTL1 (0.47) ALDH1A1THRBTHRATYMSMAPT
SCHEMBL14173224 0.80 THRB (0.45) ALDH1A1THRBTHRATYMSKDM4E
SCHEMBL8899213 0.80 MAPT (0.42) ALDH1A1THRBTHRATYMSTSHR
SCHEMBL18352540 0.80 TSHR (0.50) ALDH1A1TSHRMAPTKDM4ELMNA
SCHEMBL17708232 0.80 THRB (0.42) ALDH1A1THRBTHRATYMSTSHR
SCHEMBL27494979 0.79 THRB (0.43) PDE10AALDH1A1THRBTHRATYMS
SCHEMBL27766549 0.79 THRB (0.39) ALDH1A1THRBTHRATYMSCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233944-B1 PARTICLES FOR ELECTROPHORETIC DISPLAYS MERCK PATENT GMBH (DE) 2019-09-04 EP disclosed
EP-2393851-B1 COLOURED PARTICLES FOR ELECTROPHORETIC DISPLAYS MERCK PATENT GMBH (DE) 2018-02-28 EP disclosed
CN-102424680-A Viral polymerase inhibitors BOEHRINGER INGELHEIM CA LTD 2012-04-25 CN disclosed
CN-1558759-B Viral polymerase inhibitors BOEHRINGER INGELHEIM CA LTD 2012-01-25 CN disclosed