SCHEMBL19904576

SCHEMBL19904576

O=C(NC(Cc1cc(F)c2c(c1)OCCO2)CN1CCCC1)[C@@H]1CCN(c2ccc(Cl)c(OC3C=CC=CN3)c2)C1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 4/20 0.33
PROKR2 Q8NFJ6 3/20 0.32
HDAC4 P56524 1/20 0.32
HTR1A P08908 1/20 0.31
UGCG Q16739 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904571 0.91 PDCD1 (0.36) NOTUMHTR1AUGCGPDCD1CD274
SCHEMBL19904488 0.83 KMT2A (0.38) NOTUMPROKR2HDAC4HTR1AUGCG
SCHEMBL19904427 0.83 KMT2A (0.38) NOTUMPROKR2HDAC4HTR1AUGCG
SCHEMBL19904551 0.83 HTR1A (0.38) NOTUMPROKR2HDAC4HTR1AUGCG
SCHEMBL19904368 0.83 HTR1A (0.38) NOTUMPROKR2HDAC4HTR1AUGCG
SCHEMBL19904389 0.82 UGCG (0.40) NOTUMHTR1AUGCGPDCD1CD274
SCHEMBL19904542 0.82 UGCG (0.40) NOTUMHTR1AUGCGPDCD1CD274
SCHEMBL19904455 0.82 KMT2A (0.36) NOTUMPROKR2HTR1APDCD1CD274
SCHEMBL19904590 0.82 KMT2A (0.36) NOTUMPROKR2HTR1APDCD1CD274
SCHEMBL19904694 0.81 HTR1A (0.35) NOTUMPROKR2HTR1AUGCGPDCD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed