SCHEMBL19904694

SCHEMBL19904694

O=C(NC(Cc1cc(F)c2c(c1)OCCO2)CN1CCCC1)[C@@H]1CCN(c2ccc3cc(Cl)sc3c2)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.35
NOTUM Q6P988 4/20 0.33
TACR2 P21452 2/20 0.33
UGCG Q16739 2/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
ACACB O00763 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
CHRM2 P08172 2/20 0.31
CHRM1 P11229 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PROKR2 Q8NFJ6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904512 0.99 HTR1A (0.35) HTR1ANOTUMTACR2UGCGPDCD1
SCHEMBL19904570 0.90 NAMPT (0.33) HTR1ANOTUMUGCGPDCD1CD274
SCHEMBL19904686 0.90 NAMPT (0.33) HTR1ANOTUMUGCGPDCD1CD274
SCHEMBL19904493 0.89 KMT2A (0.38) HTR1ATACR2PDCD1CD274ACACB
SCHEMBL19904685 0.89 KMT2A (0.38) HTR1ATACR2PDCD1CD274ACACB
SCHEMBL19904427 0.88 KMT2A (0.38) HTR1ANOTUMUGCGPDCD1CD274
SCHEMBL19904455 0.87 KMT2A (0.36) HTR1ANOTUMPDCD1CD274TRPV1
SCHEMBL19904590 0.87 KMT2A (0.36) HTR1ANOTUMPDCD1CD274TRPV1
SCHEMBL19904498 0.87 KDM4E (0.37) HTR1ANOTUMUGCGACACBTRPV1
SCHEMBL19904561 0.87 MCHR1 (0.36) HTR1AUGCGCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed