SCHEMBL19904662

SCHEMBL19904662

CC(C)Oc1ccc(CC(CN2CCCC2)NC(=O)[C@@H]2CCN(c3ccc(Cl)cc3)C2)cn1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 7/20 0.43
ACACA Q13085 2/20 0.42
CCR1 P32246 1/20 0.40
HTR1A P08908 1/20 0.39
NOTUM Q6P988 1/20 0.39
TACR3 P29371 1/20 0.37
CCR5 P51681 1/20 0.37
PTGDR Q13258 1/20 0.37
TSHR P16473 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
WDR91 A4D1P6 1/20 0.36
P2RX3 P56373 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904492 0.92 ACACB (0.43) ACACBACACANOTUMTSHR
SCHEMBL19904546 0.92 ACACB (0.43) ACACBACACANOTUMTSHR
SCHEMBL19904460 0.90 ACACB (0.41) ACACBCCR1HTR1ANOTUMGPBAR1
SCHEMBL19904658 0.90 ACACB (0.41) ACACBCCR1HTR1ANOTUMGPBAR1
SCHEMBL19904665 0.88 HTR1A (0.41) CCR1HTR1ANOTUMGPBAR1
SCHEMBL19904383 0.87 ACACB (0.38) ACACBCCR1HTR1ANOTUMGPBAR1
SCHEMBL19904415 0.85 CCR1 (0.43) CCR1HTR1ANOTUMCCR5P2RX3
SCHEMBL19904651 0.85 CCR1 (0.43) CCR1HTR1ANOTUMCCR5P2RX3
SCHEMBL19904696 0.85 NOTUM (0.50) CCR1HTR1ANOTUMTSHRGPBAR1
SCHEMBL16695530 0.83 ACACB (0.46) ACACBACACACCR1NOTUMTACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed