SCHEMBL19905294

SCHEMBL19905294

CNC(=O)c1ncnc2c(C(C)[C@H](C)CNc3cc(-c4ccc(C(=O)NCCC#N)cc4)ncn3)cccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 8/20 0.40
BCR P11274 8/20 0.40
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
FAAH O00519 6/20 0.35
PRKDC P78527 2/20 0.35
ACP1 P24666 1/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CYP2D6 P10635 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17874676 0.93 ABL1 (0.41) ABL1BCRCCNB2CDK1CCNB1
SCHEMBL19905258 0.91 PRKDC (0.37) ABL1BCRFAAHPRKDC
SCHEMBL19905448 0.85 FAAH (0.47) FAAHPRKDCALDH1A1CYP1A2HSD17B10
SCHEMBL17874678 0.84 PRKDC (0.42) ABL1BCRCCNB2CDK1CCNB1
SCHEMBL15473150 0.84 PRKDC (0.42) ABL1BCRCCNB2CDK1CCNB1
SCHEMBL19905481 0.82 PRKDC (0.40) FAAHPRKDCCYP1A2CYP2D6CLK4
SCHEMBL19905365 0.81 PRKDC (0.41) FAAHPRKDC
SCHEMBL19905491 0.80 PRKDC (0.44) ABL1BCRFAAHPRKDC
SCHEMBL19905441 0.79 PRKDC (0.44) ABL1BCRFAAHPRKDCALDH1A1
SCHEMBL20415081 0.79 CCNB2 (0.34) ABL1BCRCCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057959-B1 DNA-PK INHIBITORS VERTEX PHARMA (US) 2018-02-28 EP disclosed