SCHEMBL19905896

SCHEMBL19905896

Cc1cc2nc(-c3ccnc(-c4cnc(N5CCOCC5)nc4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
CYP1A2 P05177 4/20 0.38
CASP1 P29466 4/20 0.38
CASP7 P55210 4/20 0.38
HIF1A Q16665 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP3A4 P08684 2/20 0.38
KCNH2 Q12809 2/20 0.37
PPARD Q03181 2/20 0.36
PPARA Q07869 2/20 0.36
PPARG P37231 1/20 0.35
AOC3 Q16853 1/20 0.35
USP2 O75604 3/20 0.34
HSD17B10 Q99714 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ADK P55263 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
PSEN1 P49768 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905858 0.92 USP2 (0.38) ALDH1A1CYP1A2CASP1CASP7HIF1A
SCHEMBL19906318 0.88 PPARD (0.37) KCNH2PPARDPPARAPPARGAOC3
SCHEMBL19905915 0.88 MTOR (0.40) ALDH1A1CYP1A2CASP1CASP7HIF1A
SCHEMBL19906079 0.84 ACVR1B (0.40) KCNH2
SCHEMBL19906236 0.84 PTGDR2 (0.38) ALDH1A1CYP1A2CYP2C9PPARDMEN1
SCHEMBL15341100 0.83 CYP3A4 (0.37) ALDH1A1CYP1A2CASP1CASP7HIF1A
SCHEMBL19906287 0.83 KDR (0.37) ALDH1A1MEN1KMT2APTGDR2KDM4E
SCHEMBL19906269 0.83 EIF4E (0.40) ALDH1A1CYP1A2CYP2C9PPARDMEN1
SCHEMBL19906136 0.83 GRM5 (0.36) ALDH1A1PPARDMEN1KMT2APTGDR2
SCHEMBL19905874 0.82 PTGDR2 (0.35) ALDH1A1CYP1A2CYP2C9PPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed