SCHEMBL19906079

SCHEMBL19906079

Cc1cc2nc(-c3ccnc(-c4ccc(N5CCN(C)CC5)nc4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACVR1B P36896 1/20 0.40
TGFBR1 P36897 1/20 0.40
DYRK1A Q13627 7/20 0.37
RAB9A P51151 1/20 0.37
MAPT P10636 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
MCHR1 Q99705 1/20 0.36
WNT1 P04628 4/20 0.36
GSK3B P49841 4/20 0.36
DGAT1 O75907 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH4 Q9H3N8 2/20 0.35
MET P08581 1/20 0.35
FYN P06241 1/20 0.35
MGLL Q99685 1/20 0.35
MELK Q14680 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905858 0.92 USP2 (0.38) DYRK1AMCHR1WNT1GSK3BHRH4
SCHEMBL19905818 0.91 DYRK1A (0.42) DYRK1AMAPTHTR2AHTR2CHTR2B
SCHEMBL19905854 0.90 MET (0.39) DYRK1ARAB9AMAPTHTR2AHTR2C
SCHEMBL19906164 0.88 DYRK1A (0.40) DYRK1ARAB9AMAPTHTR2AHTR2C
SCHEMBL19905981 0.86 DYRK1A (0.39) DYRK1AMAPTHTR2AHTR2CHTR2B
SCHEMBL19906287 0.85 KDR (0.37)
SCHEMBL17547119 0.84 USP2 (0.38) DYRK1AMAPTHTR2AHTR2CHTR2B
SCHEMBL19906190 0.84 MAPT (0.39) DYRK1AMAPTHTR2AHTR2CHTR2B
SCHEMBL19905896 0.84 ALDH1A1 (0.38) KCNH2
SCHEMBL19906195 0.83 CASP3 (0.37) RAB9AMAPTHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed