SCHEMBL19906269

SCHEMBL19906269

CCOc1ncc(-c2cc(-c3nc4cc(C)c(CC(=O)O)c(-c5ccc(Cl)cc5)c4s3)ccn2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF4E P06730 1/20 0.40
PTGDR2 Q9Y5Y4 6/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 3/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906236 0.93 PTGDR2 (0.38) EIF4EPTGDR2KDM4EALDH1A1MEN1
SCHEMBL19906268 0.88 EIF4E (0.38) EIF4EPTGDR2KDM4EALDH1A1MEN1
SCHEMBL19905874 0.85 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906015 0.85 PIK3CG (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906249 0.84 ALDH1A1 (0.43) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19906329 0.84 KDM4E (0.36) EIF4EPTGDR2KDM4EALDH1A1MEN1
SCHEMBL19906287 0.84 KDR (0.37) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL19905858 0.83 USP2 (0.38) PTGDR2KDM4EALDH1A1MEN1KMT2A
SCHEMBL15342614 0.83 CYP3A4 (0.38) EIF4EALDH1A1MAPTTRPM8LMNA
SCHEMBL19905939 0.83 PTGDR2 (0.35) PTGDR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed