SCHEMBL19905979

SCHEMBL19905979

Cc1cc2nc(-c3ccnc(-c4ccc5c(c4)C(=O)N(C)CCO5)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
PTGER3 P43115 3/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
KCNH2 Q12809 1/20 0.31
GPR142 Q7Z601 1/20 0.31
CPT1A P50416 2/20 0.31
CPT1B Q92523 2/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
GRM5 P41594 1/20 0.30
FFAR1 O14842 1/20 0.30
PPARD Q03181 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906111 0.92 PTGER3 (0.38) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906107 0.90 CPT1A (0.32) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19905990 0.89 GRM5 (0.39) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906136 0.88 GRM5 (0.36) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL15342612 0.84 CYP3A4 (0.36) CYP3A4
SCHEMBL19906202 0.83 PTGER3 (0.40) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL15342206 0.83 CYP3A4 (0.32) CYP3A4
SCHEMBL19906108 0.83 CPT1A (0.35) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906022 0.81 PTGER3 (0.37) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19905938 0.81 PTGDR2 (0.34) KDM4EMEN1ALDH1A1KMT2APTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed