SCHEMBL19906111

SCHEMBL19906111

Cc1cc2nc(-c3ccnc(-c4ccc5c(c4)N(C)CCO5)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 4/20 0.38
CPT1A P50416 5/20 0.34
CPT1B Q92523 5/20 0.34
PPARD Q03181 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
GRM5 P41594 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
KLKB1 P03952 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
PIK3CD O00329 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905990 0.95 GRM5 (0.39) PTGER3GRM5KDM4EMEN1ALDH1A1
SCHEMBL19905979 0.92 KDM4E (0.33) PTGER3CPT1ACPT1BPPARDGRM5
SCHEMBL19906108 0.89 CPT1A (0.35) PTGER3CPT1ACPT1BPPARDPPARG
SCHEMBL19906136 0.89 GRM5 (0.36) PTGER3CPT1ACPT1BPPARDGRM5
SCHEMBL19906202 0.88 PTGER3 (0.40) PTGER3CPT1ACPT1BKDM4EMEN1
SCHEMBL19905938 0.88 PTGDR2 (0.34) CPT1ACPT1BPPARDPPARGPPARA
SCHEMBL19906195 0.87 CASP3 (0.37) KDM4EMEN1ALDH1A1KMT2APTGDR2
SCHEMBL19906394 0.85 GRM5 (0.36) PTGER3CPT1ACPT1BPPARDGRM5
SCHEMBL19906022 0.84 PTGER3 (0.37) PTGER3CPT1ACPT1BPPARDPPARA
SCHEMBL15342615 0.83 CYP3A4 (0.37) PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed