SCHEMBL19906127

SCHEMBL19906127

Cc1cc2nc(-c3ccnc(-c4cccc5c4CCN5C)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 1/20 0.36
KDM4E B2RXH2 3/20 0.34
PTGDR2 Q9Y5Y4 3/20 0.34
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
PDE5A O76074 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE1C Q14123 1/20 0.33
PDE3A Q14432 1/20 0.33
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PPARA Q07869 4/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19906116 0.94 KMT2A (0.36) FABP4KDM4EPTGDR2ALDH1A1KMT2A
SCHEMBL19905918 0.88 PTGDR2 (0.34) FABP4KDM4EPTGDR2ALDH1A1KMT2A
SCHEMBL19906195 0.86 CASP3 (0.37) KDM4EPTGDR2ALDH1A1KMT2AMEN1
SCHEMBL19905938 0.86 PTGDR2 (0.34) KDM4EPTGDR2ALDH1A1KMT2AMEN1
SCHEMBL15342609 0.84 CYP3A4 (0.34)
SCHEMBL19906264 0.83 PTGER3 (0.34) FABP4KDM4EPTGDR2ALDH1A1KMT2A
SCHEMBL15342205 0.82 S1PR1 (0.31) S1PR1S1PR3
SCHEMBL19906111 0.82 PTGER3 (0.38) KDM4EPTGDR2ALDH1A1KMT2AMEN1
SCHEMBL19905990 0.81 GRM5 (0.39) KDM4EPTGDR2ALDH1A1KMT2AMEN1
SCHEMBL19906113 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed