SCHEMBL19906329

SCHEMBL19906329

Cc1cc2nc(-c3ccnc(-c4cncc(C(=O)O)c4)c3)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.36
PTGDR2 Q9Y5Y4 5/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAP4K4 O95819 1/20 0.34
SCN2A Q99250 2/20 0.33
SCN10A Q9Y5Y9 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
POLB P06746 1/20 0.33
KMO O15229 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
CTSA P10619 1/20 0.33
EIF4E P06730 1/20 0.33
FHIT P49789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19905772 0.94 MAP4K4 (0.41) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906328 0.87 PTGER1 (0.34) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905802 0.86 MAP4K4 (0.43) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906249 0.84 ALDH1A1 (0.43) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906236 0.84 PTGDR2 (0.38) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906247 0.84 ABL1 (0.40) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL17547144 0.84 PTGDR2 (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906269 0.84 EIF4E (0.40) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906287 0.84 KDR (0.37) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906015 0.83 PIK3CG (0.38) KDM4EPTGDR2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3070081-B1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING AN HIV INFECTION GILEAD SCIENCES INC (US) 2018-02-28 EP disclosed