SCHEMBL19916740

SCHEMBL19916740

CCC(C)c1nc2ccc(N(C)C)cc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 4/20 0.50
AAK1 Q2M2I8 2/20 0.45
ALDH1A1 P00352 2/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP1A2 P05177 1/20 0.43
TCF4 P15884 1/20 0.42
CTNNB1 P35222 1/20 0.42
APP P05067 2/20 0.41
MAPT P10636 1/20 0.41
USP2 O75604 1/20 0.41
HPGD P15428 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
PSMB5 P28074 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19132264 0.84 KDM4E (0.54) SCN10AAAK1ALDH1A1ALOX15HTT
SCHEMBL26427165 0.80 CYP1A2 (0.67) SCN10AAAK1ALDH1A1ALOX15HTT
SCHEMBL19132656 0.75 DDAH1 (0.54) ALDH1A1HTTMEN1KMT2ATCF4
SCHEMBL6367658 0.75 SCN10A (0.41) SCN10AALDH1A1ALOX15HTTMEN1
SCHEMBL1284420 0.74 TAAR1 (0.59) ALDH1A1KMT2AALPL
SCHEMBL3813964 0.74 MLKL (0.59) SCN10AALDH1A1ALOX15HTTMEN1
SCHEMBL9263421 0.74 KDM4E (0.71) SCN10AAAK1ALDH1A1ALOX15HTT
SCHEMBL23815820 0.73 SCN10A (0.71) SCN10AAAK1ALDH1A1ALOX15HTT
SCHEMBL13996322 0.73 ALDH1A1 (0.58) ALDH1A1MEN1KMT2ATCF4CTNNB1
SCHEMBL13071044 0.72 AAK1 (0.53) SCN10AAAK1ALDH1A1HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2661425-B1 HEDGEHOG ANTAGONISTS HAVING ZINC BINDING MOIETIES CURIS INC (US) 2018-02-28 EP disclosed