SCHEMBL19917535

SCHEMBL19917535

Cc1ccccc1-c1ccc2c(c1)c1ccccc1n2-c1cc(-c2ccccc2C#N)cc(-n2c3ccccc3c3cc(-c4ccccc4C)ccc32)c1C#N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.42
CYP1A2 P05177 7/20 0.38
CYP3A4 P08684 7/20 0.38
ALDH1A1 P00352 4/20 0.38
HSD17B10 Q99714 4/20 0.38
HPGD P15428 4/20 0.38
CLK4 Q9HAZ1 2/20 0.38
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 4/20 0.36
TRPA1 O75762 1/20 0.36
NR3C1 P04150 1/20 0.36
ESR2 Q92731 1/20 0.35
PPARG P37231 1/20 0.35
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
TSHR P16473 2/20 0.34
TP53 P04637 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19917534 0.97 AR (0.44) ARCYP1A2CYP3A4ALDH1A1HSD17B10
SCHEMBL19917585 0.93 TRPA1 (0.40) CYP1A2CYP3A4ALDH1A1HSD17B10HPGD
SCHEMBL22898461 0.92 TRPA1 (0.36) ARCYP1A2CYP3A4ALDH1A1HSD17B10
SCHEMBL19917533 0.90 AR (0.44) ARCYP1A2CYP3A4ALDH1A1HSD17B10
SCHEMBL19917599 0.89 PDE9A (0.35) CYP1A2CYP3A4ALDH1A1HSD17B10HPGD
SCHEMBL19917611 0.87 GABRA1 (0.37) CYP1A2CYP3A4ALDH1A1HSD17B10HPGD
SCHEMBL25660361 0.87 AR (0.45) ARALDH1A1MAPT
SCHEMBL19917536 0.87 ALDH1A1 (0.39) ARCYP1A2CYP3A4ALDH1A1HSD17B10
SCHEMBL19917552 0.87 ESR2 (0.41) CYP1A2CYP3A4ALDH1A1HSD17B10HPGD
SCHEMBL21414217 0.87 AR (0.37) ARCYP1A2CYP3A4ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504200-B1 HETEROCYCLICALLY SUBSTITUTED BIPHENYLS, ESPECIALLY FOR USE IN OPTOELECTRONIC APPARATUSES CYNORA GMBH (DE) 2021-01-20 EP disclosed
WO-2018037069-A1 HETEROCYCLICALLY SUBSTITUTED BIPHENYLS, ESPECIALLY FOR USE IN OPTOELECTRONIC APPARATUSES CYNORA GMBH (DE) 2018-03-01 WO disclosed