SCHEMBL19934868

SCHEMBL19934868

O=C(c1ccc(F)c(F)c1F)N1CC(O)C1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 3/20 0.55
MAP2K2 P36507 1/20 0.55
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
HPGD P15428 3/20 0.46
USP2 O75604 1/20 0.45
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
CPS1 P31327 5/20 0.40
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
TACR3 P29371 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4636613 0.82 CES2 (0.46) MAP2K1MAP2K2CES2CES1HPGD
SCHEMBL189188 0.73 MAP2K1 (1.00) MAP2K1MAP2K2
SCHEMBL22453383 0.73 MAP2K1 (0.76) MAP2K1MAP2K2CPS1
SCHEMBL29413551 0.73 MAP2K1 (1.00) MAP2K1MAP2K2
Hydrochloric Acid SCHEMBL29413470 0.72 MAP2K1 (0.98) MAP2K1MAP2K2
SCHEMBL23707602 0.70 MAP2K1 (0.66) MAP2K1MAP2K2CPS1
SCHEMBL30937118 0.69 HSD11B1 (0.56)
SCHEMBL4635103 0.69 P2RX7 (0.45) MAP2K1MAP2K2HPGDUSP2CPS1
SCHEMBL1760850 0.68 CES2 (0.73) MAP2K1MAP2K2CES2CES1HPGD
SCHEMBL8167393 0.68 PAX8 (0.47) MAP2K1MAP2K2CES2CES1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2909188-B1 NOVEL PROCESS FOR MAKING COMPOUNDS FOR USE IN THE TREATMENT OF CANCER EXELIXIS INC (US) 2018-03-07 EP disclosed