SCHEMBL19936632

SCHEMBL19936632

COCc1cc(-c2ccc(Cl)cc2OC)nn1C

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
CRHR1 P34998 15/20 0.42
GRM5 P41594 1/20 0.39
ADORA2B P29275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3436656 0.88 HSP90AA1 (0.46) HSP90AA1HSP90AB1CRHR1ADORA2B
SCHEMBL19936567 0.84 HSP90AA1 (0.43) HSP90AA1HSP90AB1CRHR1GRM5ADORA2B
SCHEMBL14805079 0.77 CYP1A2 (0.42) CRHR1GRM5
SCHEMBL19936425 0.77 HSP90AA1 (0.46) HSP90AA1HSP90AB1CRHR1ADORA2B
SCHEMBL19936646 0.76 CRHR1 (0.42) HSP90AA1HSP90AB1CRHR1GRM5ADORA2B
SCHEMBL14805082 0.75 HTR2A (0.45)
SCHEMBL3436592 0.75 CYP1A2 (0.44) HSP90AA1HSP90AB1CRHR1
SCHEMBL10049095 0.74 HSP90AA1 (0.43) HSP90AA1HSP90AB1CRHR1ADORA2B
SCHEMBL19936645 0.73 ESRRA (0.41) CRHR1
SCHEMBL3436659 0.72 ACHE (0.40) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2594555-B1 HETEROCYCLIC COMPOUND, AND p27 KIP1 DEGRADATION INHIBITOR ASKA PHARM CO LTD (JP) 2018-03-07 EP disclosed