SCHEMBL19953176

SCHEMBL19953176

Fc1cccc(F)c1-c1cncn1-c1ccccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.47
IDO1 P14902 4/20 0.39
TDO2 P48775 4/20 0.39
P2RX7 Q99572 1/20 0.37
KCNN4 O15554 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PDE2A O00408 1/20 0.35
PDE10A Q9Y233 1/20 0.35
HCAR1 Q9BXC0 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP3A4 P08684 1/20 0.34
MAPK14 Q16539 2/20 0.34
MAPK11 Q15759 1/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19967304 0.82 HSP90AA1 (0.49) IDO1TDO2KCNN4RAB9ATDP1
SCHEMBL19953169 0.79 CYP3A4 (0.43) GPBAR1IDO1TDO2PDE2APDE10A
SCHEMBL1076208 0.77 HSP90AA1 (0.45) IDO1TDO2RAB9ACYP11B1CYP11B2
SCHEMBL19952995 0.73 HCAR1 (0.40) KCNN4PDE2APDE10AHCAR1CYP11B2
SCHEMBL9473672 0.67 NOTUM (0.43) GPBAR1IDO1TDO2TDP1HCAR1
SCHEMBL19953054 0.67 IDO1 (0.39) IDO1TDO2
SCHEMBL19953116 0.66 HSP90AA1 (0.43) GPBAR1
SCHEMBL30349922 0.66 ALDH1A1 (0.44) GPBAR1RAB9ATDP1HCAR1
SCHEMBL19953047 0.65 HSP90AA1 (0.45) CYP11B1CYP11B2
SCHEMBL19953125 0.64 CYP11B2 (0.37) GPBAR1IDO1TDO2CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed