SCHEMBL19952995

SCHEMBL19952995

Fc1cccc(F)c1-c1c(Cl)ncn1-c1ccccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 3/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
PDE2A O00408 1/20 0.38
PDE10A Q9Y233 1/20 0.38
KCNN4 O15554 1/20 0.36
NOX4 Q9NPH5 1/20 0.36
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GRM1 Q13255 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953055 0.81 PTGS2 (0.37) PTGS1PTGS2PDE2APDE10AGABRG2
SCHEMBL19953173 0.77 PTGS2 (0.50) PTGS1PTGS2
SCHEMBL19953176 0.73 GPBAR1 (0.47) HCAR1PDE2APDE10AKCNN4CYP11B2
SCHEMBL7211112 0.67 HTT (0.56) HCAR1
SCHEMBL19953199 0.66 PTGS2 (0.49) PTGS1PTGS2
SCHEMBL19953164 0.64 CYP11B2 (0.47) PTGS1PTGS2CYP11B2
SCHEMBL1073380 0.64 PTGS2 (0.50) PTGS1PTGS2
SCHEMBL10593949 0.64 MAPK14 (0.42) PDE2APDE10AKCNN4
SCHEMBL10593745 0.64 MAPK14 (0.42) PDE2APDE10AKCNN4
SCHEMBL1074163 0.63 PTGS2 (0.42) PTGS1PTGS2GRM1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed