SCHEMBL19953371

SCHEMBL19953371

CCOC(=O)CCC(=O)Nc1c(C)cccc1C(N)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 4/20 0.50
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
USP2 O75604 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPT P10636 5/20 0.44
LMNA P02545 4/20 0.44
TDP1 Q9NUW8 1/20 0.44
PARP1 P09874 1/20 0.43
SCN3A Q9NY46 2/20 0.43
MEN1 O00255 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29902998 0.83 HDAC3 (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL20339486 0.83 HDAC3 (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL163242 0.81 GPR35 (0.52) NLRP3MAPTALDH1A1CYP3A4L3MBTL1
SCHEMBL25195550 0.77 POLB (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL25556173 0.77 ALDH1A1 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL31058474 0.77 ALDH1A1 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL6887530 0.75 NLRP3 (0.67) NLRP3HDAC3HDAC4HDAC1HDAC7
SCHEMBL1491077 0.75 NLRP3 (0.70) NLRP3HDAC3HDAC4HDAC1HDAC7
SCHEMBL30409645 0.75 DRD2 (0.51) LMNAPARP1MEN1KMT2AALDH1A1
SCHEMBL22426563 0.73 TSHR (0.54) NLRP3HSD17B10MAPTLMNASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018046933-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2018-03-15 WO disclosed