SCHEMBL19953603

SCHEMBL19953603

CS(=O)(=O)c1ccc(-n2ccnc2C(F)(F)F)cc1-c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.41
PTGS1 P23219 2/20 0.41
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
MAOA P21397 2/20 0.38
LOXL2 Q9Y4K0 2/20 0.38
LOX P28300 1/20 0.38
MITF O75030 1/20 0.37
LMNA P02545 1/20 0.37
STAT3 P40763 1/20 0.37
STAT1 P42224 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TLR9 Q9NR96 1/20 0.37
NR3C2 P08235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25382278 0.75 NOTUM (0.39) PTGS2PTGS1ALDH1A1SMN1; SMN2LMNA
SCHEMBL7865578 0.72 ALOX5AP (0.50) PTGS2KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL8801286 0.69 ALDH1A1 (0.37) PTGS2ALDH1A1SMN1; SMN2LMNANR3C2
SCHEMBL27454511 0.67 PTGS2 (0.51) PTGS2MAOALOXL2LOX
SCHEMBL8758545 0.65 FGFR1 (0.45) PTGS2PTGS1KDM4EALDH1A1RAB9A
SCHEMBL28003240 0.65 MAPT (0.46) HPGD
SCHEMBL8814075 0.63 CYP17A1 (0.38) PTGS2KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL31138150 0.63 PTGS2 (0.34) PTGS2KDM4E
SCHEMBL28003186 0.63 NR1I2 (0.48) PTGS2PTGS1ALDH1A1RAB9ANPC1
SCHEMBL9080396 0.62 ALDH1A1 (0.45) PTGS2PTGS1KDM4EALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049014-A1 DASH INHIBITORS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE (US) 2018-03-15 WO disclosed
CN-100457183-C Cyclooxygenase-2 inhibitor/histone deacetylase inhibitor combination NOVARTIS AG (CH) 2009-02-04 CN disclosed
CN-1578674-A Cyclooxygenase-2 inhibitor/histone deacetylase inhibitor combination NOVARTIS AG (CH) 2005-02-09 CN disclosed