SCHEMBL9080396

SCHEMBL9080396

COc1ccc(-n2ccnc2C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.42
PTGS1 P23219 3/20 0.41
PTGS2 P35354 3/20 0.41
AHR P35869 1/20 0.41
SCN5A Q14524 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP19A1 P11511 1/20 0.41
TSHR P16473 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 2/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28714521 0.85 HTT (0.43) ALDH1A1KMT2AHTTCYP1A2CYP2C9
SCHEMBL28442535 0.81 P2RX7 (0.44) ALDH1A1KMT2AKDM4EMEN1HPGD
SCHEMBL25382278 0.80 NOTUM (0.39) ALDH1A1PTGS1PTGS2SCN5ATP53
SCHEMBL28003186 0.78 NR1I2 (0.48) ALDH1A1KMT2AMEN1PTGS1PTGS2
SCHEMBL3967152 0.78 L3MBTL1 (0.50) ALDH1A1KMT2AHTTCYP1A2CYP2C9
SCHEMBL28354722 0.77 NOTUM (0.42) ALDH1A1KMT2AMEN1PTGS2CYP19A1
SCHEMBL8149329 0.77 PTGS2 (0.42) ALDH1A1KDM4EHPGDHTTPTGS1
SCHEMBL10902105 0.76 CYP3A4 (0.66) ALDH1A1KMT2AKDM4EMEN1HPGD
SCHEMBL8511275 0.75 HTT (0.45) ALDH1A1KMT2AHTTPTGS1PTGS2
SCHEMBL17844189 0.75 MAPT (0.50) ALDH1A1KMT2AMEN1HTTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1660816-A Method for synthesizing 2-perfluoroalkyl group substituted ramification of imidazole UNIV SHANGHAI (CN) 2005-08-31 CN disclosed
WO-1996003387-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed