SCHEMBL19960686

SCHEMBL19960686

COC1c2ccccc2CC1NC(=O)C1c2ccccc2CCN1C(=O)C1CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
F11 P03951 5/20 0.48
HSD11B1 P28845 2/20 0.39
OPRM1 P35372 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ACE P12821 2/20 0.37
KLKB1 P03952 2/20 0.37
TSHR P16473 1/20 0.37
XIAP P98170 2/20 0.36
CASP3 P42574 1/20 0.36
CASP2 P42575 1/20 0.36
MTNR1B P49286 2/20 0.36
DRD1 P21728 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953575 0.89 ACE (0.41) F11ACEKLKB1XIAPCASP3
SCHEMBL19953576 0.89 ACE (0.41) F11ACEKLKB1XIAPCASP3
SCHEMBL19953578 0.89 ACE (0.41) F11ACEKLKB1XIAPCASP3
SCHEMBL19960811 0.85 GHSR (0.45) XIAP
SCHEMBL19953493 0.84 F11 (0.53) F11ALDH1A1NPSR1ACEKLKB1
SCHEMBL19960718 0.83 ACE (0.46) F11ACEXIAPCASP3CASP2
SCHEMBL19960651 0.82 F11 (0.45) F11HSD11B1ALDH1A1NPSR1XIAP
SCHEMBL19960692 0.81 ACE (0.44) F11NPSR1ACECASP3CASP2
SCHEMBL19953782 0.80 F11 (0.55) F11ALDH1A1NPSR1ACEKLKB1
SCHEMBL19953516 0.79 F11 (0.53) F11HSD11B1ALDH1A1NPSR1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed