SCHEMBL19960922

SCHEMBL19960922

NC(=O)C1c2ccccc2CC(=O)N1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MEN1 O00255 1/20 0.43
APAF1 O14727 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
EHMT2 Q96KQ7 1/20 0.42
GRM7 Q14831 1/20 0.42
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
PARP1 P09874 1/20 0.40
ACE P12821 2/20 0.39
SIRT1 Q96EB6 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
CAPN1 P07384 1/20 0.38
POLB P06746 1/20 0.38
CACNA1G O43497 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953490 0.89 ACE (0.46) CYP2C9CYP2C19MEN1APAF1ALDH1A1
SCHEMBL19953697 0.89 ACE (0.46) CYP2C9CYP2C19MEN1APAF1ALDH1A1
SCHEMBL19960921 0.83 GRM7 (0.42) CYP2C9CYP2C19MEN1APAF1ALDH1A1
SCHEMBL19960416 0.81 GRM7 (0.60) GRM7OPRM1OPRK1OPRL1PARP1
SCHEMBL19960674 0.78 PARP1 (0.41) CYP2C9ALDH1A1MAPTHPGDGRM7
SCHEMBL11472266 0.74 GRIN1 (0.50) PARP1ACEGRIN1GRIN2BSIGMAR1
SCHEMBL19960826 0.73 ACE (0.47) GRM7ACE
SCHEMBL19953701 0.73 ACE (0.47) GRM7ACE
SCHEMBL19953623 0.72 L3MBTL1 (0.46) MEN1ALDH1A1MAPTKMT2AGRM7
SCHEMBL19953612 0.72 L3MBTL1 (0.46) MEN1ALDH1A1MAPTKMT2AGRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed