SCHEMBL19964625

SCHEMBL19964625

C=C(c1c(C)c(C(=O)OC(C)C)cc2cc(-c3cccc(C#N)c3)cn12)N1CCOCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.36
ALDH1A1 P00352 2/20 0.35
CNR1 P21554 1/20 0.34
EED O75530 1/20 0.34
RBBP4 Q09028 1/20 0.34
SUZ12 Q15022 1/20 0.34
EZH2 Q15910 1/20 0.34
AEBP2 Q6ZN18 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
SLC2A1 P11166 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MGLL Q99685 1/20 0.33
KCNH2 Q12809 2/20 0.33
PIK3CA P42336 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
LRRK2 Q5S007 2/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21157283 0.88 ALOX15 (0.41) ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL21113144 0.87 RAB9A (0.42) PRKDCALDH1A1L3MBTL1KDM4ESMN1; SMN2
SCHEMBL21157331 0.87 EED (0.46) PRKDCALDH1A1EEDRBBP4SUZ12
SCHEMBL28886523 0.85 EZH2 (0.42) PRKDCALDH1A1CNR1EZH2HRH2
SCHEMBL21251228 0.85 CNR2 (0.38) ALDH1A1EEDRBBP4SUZ12EZH2
SCHEMBL21156100 0.83 ALDH1A1 (0.42) ALDH1A1KDM4E
SCHEMBL21157291 0.83 EED (0.43) PRKDCALDH1A1EEDRBBP4SUZ12
SCHEMBL21156531 0.83 ALDH1A1 (0.40) ALDH1A1EEDRBBP4SUZ12EZH2
SCHEMBL21157327 0.82 PRKCZ (0.42) ALDH1A1L3MBTL1KDM4ETRPV1LMNA
SCHEMBL19964426 0.82 NPC1 (0.41) ALDH1A1KDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3524602-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Haihe Pharmaceutical Co., Ltd. (CN) 2019-08-14 EP disclosed
WO-2018045971-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海海和药物研究开发有限公司 2018-03-15 WO disclosed