SCHEMBL19968019

SCHEMBL19968019

Cc1nc(Cl)ccc1C(=O)N1CCC(=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.40
THRB P10828 1/20 0.37
HPGD P15428 4/20 0.37
USP2 O75604 1/20 0.37
RAB9A P51151 1/20 0.36
TP53 P04637 2/20 0.36
MDM2 Q00987 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SPR P35270 1/20 0.36
HTT P42858 3/20 0.36
LMNA P02545 2/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29405584 1.00 HSP90AA1 (0.40) HSP90AA1THRBHPGDUSP2RAB9A
SCHEMBL22650459 0.75 GSK3B (0.36) SPRTRPV4
SCHEMBL440559 0.75 HSP90AA1 (0.42) HSP90AA1THRBSMN1; SMN2LMNATRPV4
SCHEMBL19968008 0.74 MEN1 (0.59) TP53SPRLMNAMEN1KMT2A
SCHEMBL28731677 0.72 PDE10A (0.35) HPGDMEN1KMT2ATRPV4ALDH1A1
SCHEMBL20150154 0.71 GABRP (0.57) HPGDUSP2HTTLMNATSHR
SCHEMBL1929985 0.70 HTT (0.70) HPGDHTTKMT2AALDH1A1CYP3A4
SCHEMBL12410963 0.70 SMN1; SMN2 (0.54) RAB9AMDM2SMN1; SMN2LMNAMEN1
SCHEMBL403869 0.70 GABRP (0.46) RAB9ASMN1; SMN2ALOX15MEN1KMT2A
SCHEMBL30996511 0.70 SMN1; SMN2 (0.54) RAB9AMDM2SMN1; SMN2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120040446-A CDK inhibitors 基因泰克公司 2025-05-27 CN disclosed
US-20220296595-A1 CDK INHIBITORS GENENTECH, INC. 2022-09-22 US disclosed
CN-112225724-B Benzimidazole compound kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-04-29 CN disclosed
CN-114364675-A CDK inhibitors 上海齐鲁锐格医药研发有限公司 2022-04-15 CN disclosed
EP-3966213-A1 CDK INHIBITORS Qilu Regor Therapeutics Inc. (CN) 2022-03-16 EP disclosed
CN-112250669-B Benzimidazole compound kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-02-25 CN disclosed
CN-112250669-A Benzimidazole compound kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2021-01-22 CN disclosed
CN-112225724-A Benzimidazole compound kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2021-01-15 CN disclosed
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed
CN-109963842-B Benzimidazole compound kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2020-11-03 CN disclosed
CN-109963842-A Benzimidazoles compound kinase inhibitor and its preparation method and application 江苏豪森药业集团有限公司 2019-07-02 CN disclosed
WO-2018045956-A1 BENZIMIDAZOLE COMPOUND KINASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed
CN-107793399-A CDK4/6 inhibitor and its preparation method and application 上海翰森生物医药科技有限公司 2018-03-13 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220296595-A1 CDK INHIBITORS CDKL1, CDK9, CDK6 HSP90AA1 3152/4885THRB 3558/4885HPGD 2238/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.