SCHEMBL19971355

SCHEMBL19971355

CNC(=O)OCc1cn(S(=O)(=O)c2cccc(C(F)(F)F)c2)c2cc(N(C)c3ccc(OC)nc3Cl)ccc12

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.38
HTR6 P50406 6/20 0.34
ADORA2A P29274 2/20 0.33
ADORA2B P29275 2/20 0.33
ADORA1 P30542 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 1/20 0.33
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
HDAC6 Q9UBN7 2/20 0.32
KMT2A Q03164 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16626667 0.89 RORC (0.37) RORCHTR6ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL16619121 0.88 RORC (0.37) RORCHTR6ADORA2AADORA2BADORA1
SCHEMBL16619178 0.87 RORC (0.40) RORCHTR6ADORA2AADORA2BADORA1
SCHEMBL19971369 0.85 RORC (0.39) RORCHTR6PPARG
SCHEMBL16626662 0.84 RORC (0.37) RORCHTR6ADORA2AADORA2BADORA1
SCHEMBL16626655 0.74 RORC (0.39) RORCHTR6L3MBTL1ALDH1A1KMT2A
SCHEMBL16619006 0.74 RORC (0.40) RORCHTR6L3MBTL1ALDH1A1HDAC6
SCHEMBL16618638 0.73 HTR6 (0.42) RORCHTR6L3MBTL1ALDH1A1HDAC6
Hydrochloric Acid SCHEMBL16618977 0.73 RORC (0.39) RORCHTR6L3MBTL1KMT2A
SCHEMBL16626748 0.73 RORC (0.38) RORCHTR6L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed