SCHEMBL16626667

SCHEMBL16626667

CNCc1cn(S(=O)(=O)c2cccc(C(F)(F)F)c2)c2cc(N(C)c3ccc(OC)nc3Cl)ccc12

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.37
HTR6 P50406 14/20 0.37
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16619121 0.99 RORC (0.37) RORCHTR6ALDH1A1L3MBTL1ADORA2A
SCHEMBL19971355 0.89 RORC (0.38) RORCHTR6ALDH1A1L3MBTL1ADORA2A
SCHEMBL16619178 0.88 RORC (0.40) RORCHTR6ALDH1A1L3MBTL1ADORA2A
SCHEMBL16626662 0.85 RORC (0.37) RORCHTR6ALDH1A1L3MBTL1ADORA2A
SCHEMBL16626655 0.85 RORC (0.39) RORCHTR6ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL16618977 0.84 RORC (0.39) RORCHTR6L3MBTL1
SCHEMBL16626748 0.83 RORC (0.38) RORCHTR6ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL16618931 0.83 RORC (0.38) RORCHTR6ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL16618681 0.77 RORC (0.38) RORCHTR6ALDH1A1L3MBTL1
SCHEMBL16618638 0.77 HTR6 (0.42) RORCHTR6ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP claimed
EP-3052484-B1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAE WOONG PHARMA (KR) 2018-03-21 EP disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-9676714-B2 Sulfonylindole derivatives and method for preparing the same DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2017-06-13 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2016-08-04 US disclosed
WO-2015050412-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221946-A1 SULFONYLINDOLE DERIVATIVES AND METHOD FOR PREPARING THE SAME GIPR, PGC, SI RORC 1067/4885HTR6 166/4885ALDH1A1 2153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.