SCHEMBL19975167

SCHEMBL19975167

Cc1cnc([C@@H](CNC(=O)O)c2ccc(OCc3ccccc3)cc2)o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.47
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
PKM P14618 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
P4HTM Q9NXG6 1/20 0.44
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
CASP3 P42574 1/20 0.44
HTT P42858 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
ALOX5 P09917 1/20 0.44
ACACB O00763 1/20 0.43
MAOB P27338 1/20 0.43
FFAR1 O14842 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3550137 0.86 FFAR1 (0.53) IDH1P4HTMLMNAGAAHPGD
SCHEMBL13550298 0.83 IDH1 (0.47) IDH1MAPTRAB9ASMN1; SMN2P4HTM
SCHEMBL3517268 0.83 LMNA (0.49) IDH1ALDH1A1P4HTMLMNAGAA
SCHEMBL13140162 0.82 IDH1 (0.47) IDH1NPC1ALDH1A1MAPTPKM
Hydrochloric Acid SCHEMBL19974577 0.81 MAOB (0.47) IDH1MAPTRAB9ASMN1; SMN2LMNA
SCHEMBL23296263 0.78 PPARG (0.47) NPC1ALDH1A1MAPTPKMRAB9A
SCHEMBL23296264 0.78 PPARG (0.47) NPC1ALDH1A1MAPTPKMRAB9A
SCHEMBL20425199 0.76 NR4A1 (0.53) LMNAALOX5ACACBMAOBFFAR1
SCHEMBL25922304 0.74 SIGMAR1 (0.46) IDH1LMNAMAOBL3MBTL1
SCHEMBL19982217 0.73 LTA4H (0.51) IDH1MAPTRAB9ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512839-A1 YAP1 INHIBITORS THAT TARGET THE INTERACTION OF YAP1 WITH OCT4 H. Lee Moffitt Cancer Center And Research Institute, Inc. (US) 2019-07-24 EP disclosed
WO-2018053446-A1 YAP1 INHIBITORS THAT TARGET THE INTERACTION OF YAP1 WITH OCT4 H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2018-03-22 WO disclosed