SCHEMBL20425199

SCHEMBL20425199

O=C(O)NC[C@H](O)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.53
NR4A2 P43354 1/20 0.53
NR4A3 Q92570 1/20 0.53
MAOB P27338 1/20 0.50
PARP10 Q53GL7 1/20 0.50
ALOX5 P09917 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
PTGS1 P23219 1/20 0.50
SLC6A2 P23975 1/20 0.50
CYP2C19 P33261 1/20 0.50
PTGS2 P35354 1/20 0.50
SLC6A3 Q01959 1/20 0.50
HIF1A Q16665 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
ACACB O00763 1/20 0.49
FFAR1 O14842 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL323396 0.87 LTA4H (0.48) NR4A1NR4A2NR4A3MAOBALOX5
SCHEMBL3837460 0.87 FFAR1 (0.51) MAOBALOX5ACACBFFAR1
SCHEMBL15232863 0.85 KMT2A (0.57) NR4A2MAOBALOX5
SCHEMBL1553476 0.83 SYK (0.54) MAOBALOX5ACACB
SCHEMBL2295812 0.82 HIF1A (0.56) MAOBALOX5LMNACYP1A2PTGS1
SCHEMBL2296971 0.82 HIF1A (0.56) MAOBALOX5LMNACYP1A2PTGS1
SCHEMBL9537619 0.82 GSK3B (0.49) NR4A1NR4A2NR4A3MAOBPARP10
SCHEMBL20425137 0.82 PPARG (0.59) NR4A1NR4A2NR4A3MAOBFFAR1
SCHEMBL19974547 0.81 FFAR1 (0.54) NR4A1NR4A2NR4A3MAOBALOX5
SCHEMBL323593 0.81 BCHE (0.64) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018138739-A1 NOVEL ANTIESTROGENIC HETEROCYCLIC COMPOUNDS SUN PHARMA ADVANCED RESEARCH COMPANY LIMITED (IN) 2018-08-02 WO disclosed