SCHEMBL19980227

SCHEMBL19980227

CNC(=O)/C(N)=C/NCc1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
RAB9A P51151 2/20 0.45
MAPT P10636 1/20 0.45
GLA P06280 1/20 0.45
KDM4E B2RXH2 2/20 0.42
HPGD P15428 4/20 0.41
LMNA P02545 2/20 0.41
KMT2A Q03164 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20344664 0.84 ADH1B (0.46) ALDH1A1RAB9AMAPTKDM4EHPGD
SCHEMBL21156962 0.84 ALDH1A1 (0.46) ALDH1A1RAB9AMAPTGLAKDM4E
SCHEMBL21156950 0.71 ALDH1A1 (0.46) ALDH1A1RAB9AMAPTGLAKDM4E
SCHEMBL24247846 0.70 ALDH1A1 (0.45) ALDH1A1RAB9AMAPTGLAKDM4E
SCHEMBL17261148 0.70 PLA2G1B (0.47) ALDH1A1RAB9AMAPTGLAHPGD
SCHEMBL7950040 0.68 RAB9A (0.60) ALDH1A1RAB9AHPGDLMNAKMT2A
SCHEMBL689542 0.68 CYP2C19 (0.66) ALDH1A1RAB9AHPGDLMNAKMT2A
SCHEMBL7449229 0.67 ADH1B (0.52) ALDH1A1RAB9AMAPTHPGDLMNA
SCHEMBL7449222 0.67 ADH1B (0.52) ALDH1A1RAB9AMAPTHPGDLMNA
SCHEMBL20344487 0.67 ADH1B (0.52) ALDH1A1RAB9AMAPTHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3342771-A1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GlaxoSmithKline Intellectual Property Development Ltd (GB) 2018-07-04 EP disclosed
EP-2956452-B1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2018-03-21 EP disclosed