SCHEMBL19980475

SCHEMBL19980475

Bc1ccc2c3c(cccc13)C1(c3ccccc3-c3ccccc31)c1ccccc1-2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
OPRK1 P41145 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 2/20 0.32
TSHR P16473 2/20 0.32
MAPK1 P28482 2/20 0.32
HSD17B10 Q99714 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
HIF1A Q16665 1/20 0.32
PABPC1 P11940 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19980463 0.87 MAOA (0.33) PDK2
SCHEMBL12337351 0.82 CRHBP (0.39) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL23430646 0.80 KEAP1 (0.63) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL30343464 0.80 CYP1A2 (0.47) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL19980414 0.80 CYP1A2 (0.47) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL2723227 0.78 KDM4E (0.42) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL9613694 0.78 KEAP1 (0.58) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL19974226 0.76 ESR1 (0.34) CRHBPCRHR2KEAP1NFE2L2KDM4E
SCHEMBL29516015 0.74 ALDH1A1 (0.54) CRHBPCRHR2KDM4EMAPTSMN1; SMN2
SCHEMBL19974426 0.74 ALDH1A1 (0.54) CRHBPCRHR2KDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512841-B1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES MERCK PATENT GMBH (DE) 2023-04-26 EP disclosed
WO-2018050584-A1 COMPOUNDS WITH SPIROBIFLUORENE-STRUCTURES MERCK PATENT GMBH (DE) 2018-03-22 WO disclosed