SCHEMBL19981328

SCHEMBL19981328

C=C(C(N)=O)[C@H](NS(=O)(=O)N1CCOCC1)c1nc(-c2cnccn2)no1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 1/20 0.36
PKM P14618 2/20 0.34
GAA P10253 1/20 0.34
POLB P06746 1/20 0.34
EPHX2 P34913 1/20 0.33
KCNH2 Q12809 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ATM Q13315 1/20 0.33
ALDH1A1 P00352 1/20 0.33
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
GSK3B P49841 4/20 0.33
DYRK1A Q13627 4/20 0.33
KDM4E B2RXH2 1/20 0.32
CCNE2 O96020 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19981270 0.83 BMP1 (0.40) BMP1PKMGAAPOLBEPHX2
SCHEMBL19981170 0.79 BMP1 (0.36) BMP1PKMPOLBEPHX2KCNH2
SCHEMBL19981267 0.76 BMP1 (0.34) BMP1PKMKDM4ENPC1RAB9A
SCHEMBL19981266 0.71 BMP1 (0.37) BMP1PKMPOLBEPHX2KCNH2
SCHEMBL19984850 0.68 HDAC6 (0.40) PKMGAAPOLBGSK3BDYRK1A
SCHEMBL19981145 0.67 BMP1 (0.49) BMP1PKMEPHX2KCNH2TDP1
SCHEMBL19981325 0.65 BMP1 (0.38) BMP1PKMPOLBEPHX2KCNH2
SCHEMBL19981138 0.64 BMP1 (0.49) BMP1PKMEPHX2KCNH2TDP1
SCHEMBL18078059 0.63 BMP1 (0.46) BMP1PKMPOLBTDP1ATM
SCHEMBL19981324 0.63 BMP1 (0.36) BMP1PKMPOLBTDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051254-A1 CYCLIC SUBSTITUTED-1,2,4-OXADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed