SCHEMBL19984850

SCHEMBL19984850

NC(=O)C[C@H](NS(=O)(=O)N1CCOCC1)c1nnc(-c2cnccn2)o1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 8/20 0.40
LRRK2 Q5S007 1/20 0.36
HDAC1 Q13547 2/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
NAMPT P43490 1/20 0.33
GAA P10253 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19981270 0.83 BMP1 (0.40) LRRK2POLBPKMMAPTHTT
SCHEMBL19984831 0.83 LRRK2 (0.35) HDAC6LRRK2HDAC1POLBPKM
SCHEMBL19984824 0.77 HDAC6 (0.34) HDAC6NAMPTCYP2C9CYP2C19
SCHEMBL19984805 0.73 NPY5R (0.37) HDAC6LRRK2POLBPKMMAPT
SCHEMBL18078725 0.69 CD274 (0.52) POLB
SCHEMBL19866357 0.69 CD274 (0.52) POLB
SCHEMBL19984975 0.69 TRHR (0.36) MAPT
SCHEMBL19973939 0.69 MAPK1 (0.33) POLB
SCHEMBL19973940 0.69 MAPK1 (0.33) POLB
SCHEMBL19981328 0.68 BMP1 (0.36) LRRK2POLBPKMMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051255-A1 CYCLIC SUBSTITUTED-1,3,4-OXADIAZOLE AND THIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed