SCHEMBL1998156

SCHEMBL1998156

Clc1cccc(-c2c(-c3ccnc(Cl)c3)[nH]c3nccnc23)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.46
MAPK14 Q16539 3/20 0.46
MAPK13 O15264 2/20 0.46
MAPK12 P53778 2/20 0.46
MAPK11 Q15759 2/20 0.46
NUDT1 P36639 5/20 0.43
CCNB2 O95067 3/20 0.41
CDK1 P06493 3/20 0.41
CCNB1 P14635 3/20 0.41
GSK3A P49840 3/20 0.41
GSK3B P49841 3/20 0.41
CCNB3 Q8WWL7 3/20 0.41
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
LRRK2 Q5S007 2/20 0.39
PTGS2 P35354 1/20 0.38
NPY5R Q15761 1/20 0.38
STK4 Q13043 1/20 0.38
STK3 Q13188 1/20 0.38
GRIN2D O15399 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999001 0.81 MAPK14 (0.69) METMAPK14MAPK13MAPK12MAPK11
SCHEMBL1997010 0.79 MAPK14 (0.42) METMAPK14MAPK13MAPK12MAPK11
SCHEMBL2286613 0.70 MET (0.67) METMAPK14MAPK13MAPK12MAPK11
SCHEMBL2785987 0.69 MAPK14 (0.73) METMAPK14MAPK13MAPK12MAPK11
SCHEMBL13379720 0.68 MAPK14 (0.45) MAPK14MAPK13MAPK12MAPK11CCNB2
SCHEMBL1996761 0.68 MAPK14 (0.51) METMAPK14MAPK13MAPK12MAPK11
SCHEMBL2125635 0.67 IDO1 (0.47) MAPK14MAPK13MAPK12MAPK11NUDT1
SCHEMBL2886849 0.66 MAPK14 (0.70) METMAPK14MAPK13MAPK12MAPK11
SCHEMBL26910396 0.65 TGFBR1 (0.40) CCNB2CDK1CCNB1CCNB3CDK5
SCHEMBL2786751 0.65 CCNB2 (0.49) MAPK14MAPK13MAPK12MAPK11CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2338890-A1 4,7-Diazaindole derivatives and their use as fungicides Bayer CropScience AG (DE) 2011-06-29 EP claimed
WO-2010046215-A2 DIAZA-INDOLE DERIVATIVES AND THEIR USE AS FUNGICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-04-29 WO claimed
EP-2338890-A1 4,7-Diazaindole derivatives and their use as fungicides Bayer CropScience AG (DE) 2011-06-29 EP disclosed
WO-2010046215-A2 DIAZA-INDOLE DERIVATIVES AND THEIR USE AS FUNGICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-04-29 WO disclosed