SCHEMBL19981565

SCHEMBL19981565

Cc1c(C(=N)/C=C(/Nc2cc(C)n(C)n2)C(N)=O)ccc(F)c1N

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
CHRM4 P08173 2/20 0.34
HDAC6 Q9UBN7 1/20 0.32
MAP3K5 Q99683 1/20 0.31
GRM5 P41594 1/20 0.31
BACE1 P56817 1/20 0.30
CHKA P35790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19981750 0.78 BTK (0.37) HDAC6
SCHEMBL19981966 0.78 BTK (0.37) HDAC6
SCHEMBL19981813 0.77 BTK (0.36) LMNA
SCHEMBL19981978 0.77 BTK (0.32)
SCHEMBL19981793 0.76 CLK1 (0.42)
SCHEMBL19981564 0.76 KDM4E (0.31) ALDH1A1
SCHEMBL12025148 0.73 BTK (0.43) CHRM4
SCHEMBL19981725 0.67 BTK (0.45) HDAC6
SCHEMBL10274568 0.65 ALDH1A1 (0.63) ALDH1A1LMNAMAP3K5CHKA
SCHEMBL26847445 0.64 SMN1; SMN2 (0.56) ALDH1A1LMNAMAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2365970-B1 PYRIDAZINONES AND THEIR USE AS BTK INHIBITORS GILEAD CONNECTICUT INC (US) 2018-03-21 EP disclosed