SCHEMBL1998318

SCHEMBL1998318

O=C(c1cnc(-c2cccnc2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.44
HDAC1 Q13547 3/20 0.43
ALDH1A1 P00352 6/20 0.41
KDM4E B2RXH2 4/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
PTGES2 Q9H7Z7 2/20 0.40
HDAC8 Q9BY41 1/20 0.39
LMNA P02545 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004973 0.92 PTGES2 (0.42) HDAC6HDAC1ALDH1A1KDM4EHPGD
SCHEMBL2002616 0.91 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTCYP1A2CYP3A4
SCHEMBL2008737 0.90 LMNA (0.42) HDAC6HDAC1ALDH1A1KDM4EHPGD
SCHEMBL2003496 0.90 ALDH1A1 (0.40) HDAC6HDAC1ALDH1A1KDM4ECYP1A2
SCHEMBL2003239 0.90 PTGES2 (0.41) HDAC6HDAC1ALDH1A1KDM4EHPGD
SCHEMBL2002956 0.89 PTGES2 (0.44) HDAC6HDAC1ALDH1A1KDM4EHPGD
SCHEMBL2007614 0.88 PTGES2 (0.41) HDAC6HDAC1ALDH1A1KDM4EHPGD
SCHEMBL1999932 0.88 RAB9A (0.46) HDAC6HDAC1ALDH1A1KDM4EHPGD
SCHEMBL2002482 0.87 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL2002164 0.86 ALOX5AP (0.45) HDAC6HDAC1ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed